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AM-1221 Powder 100g

AM-1221 Powder 100g

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AM-1221 Powder

AM-1221 is a drug that acts as a potent and selective agonist for the cannabinoid receptor CB2, with a Ki of 0.28nM at CB2 and 52.3nM at the CB1 receptor, giving it around 180x selectivity for CB2.The 2-methyl and 6-nitro groups on the indole ring both tend to increase CB2 affinity while generally reducing affinity at CB1, explaining the high CB2 selectivity of AM-1221. However despite this relatively high selectivity for CB2, its CB1 affinity is still too strong to make it useful as a truly selective CB2 agonist, so the related compound AM-1241 is generally preferred for research purposes.

AM-1221

IUPAC name: 1-[(N-methylpiperidin-2-yl)methyl]-2-methyl-3-(naphthalen-1-oyl)-6-nitroindole

CAS number: 335160-53-7

Formula: C27H27N3O3

Purity: 99,6% min

Appearance: white powder

AM-1221 is a chemical for research purposes and should only be used for this purpose. AM-2201 is not sold for human consumption.

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